Ulwazi Lomkhiqizo
Ukwethulwa kwe-cepharanthine
I-cepharanthine iyi-benzyl isowaline alkaloid enama-benzyl amabili ehlukanisiwe futhi ekhishwe ezitshalweni ze-tetragoniaceae. Inemisebenzi yokulawula isimila, i-anti-malarial, i-antibacterial, kanye ne-immune function regulation. Ucwaningo lwanamuhla lusikisela ukuthi luphinde lube nemisebenzi yokuvuselela i-reticuloendothelial uhlelo, ukuvuselela izicubu ze-hematopoietic, nokukhuthaza ukwanda kwezicubu zomnkantsha wamathambo.Ngakho-ke, i-cepharanthine ibhekwa njengesidakamizwa esinobuthi obuphansi futhi esisebenzayo sokukhulisa i-leukocyte.Njengamanje, ososayensi baseChina bathole ukuthi inani elincane kakhulu le-cepharanthine lingavimba ukwanda nokusabalala kwe-coronavirus entsha.
indima cepharanthine
I-Chrysanthemum inomphumela we-antitumor ongase ube namandla.Ukusetshenziswa okukodwa kwe-cepharanthine kungadlala umphumela wokulwa nesimila ngokuvimbela ukwanda kwamangqamuzana esimila kanye nokuthuthukisa ukuzivikela komzimba.Okuthembisa kakhulu ukuthi i-cepharanthine ehlanganiswe nemithi yokwelapha ingakwazi ukuthuthukisa ukusebenza kahle kwe-chemotherapy ngokunciphisa ukumelana nezidakamizwa kwamangqamuzana.Indlela eyinhloko ingase ibe ukuthi i-cepharanthine ingakhuphula ukunqwabelana kwezidakamizwa ezilwa nomdlavuza emangqamuzaneni ngokuphazamisa umsebenzi we-plasma membrane.Ngaphezu kwalokho, i-cepharanthine ingaphinde ithuthukise ukuzwela kwamangqamuzana e-tumor ku-radiotherapy.I-anti-Direct anti- umphumela wesimila we-cepharanthine:i-cepharanthine ingathuthukisa ikhono lomzimba lokulwa ne-tumor ngokuthuthukisa ukusabela komzimba komzimba.Ama-Macrophage angakwazi ukubona ngokuqondile futhi abulale amangqamuzana e-tumor futhi adlale indima ebalulekile ekuvikelekeni kwe-tumor.Kodwa-ke, kubantu abane-tumorigenesis, ama-macrophages avame ivinjiwe.I-Chrysanthin ingenza kusebenze ama-macrophage, okungenzeka ahlobane nomthelela wawo ekwelapheni kwesimila.
NgoMeyi 10,2022, umuthi omusha wokwelapha i-COVID-19 otholwe ososayensi baseShayina wanikezwa ilungelo lobunikazi lokusungulwa kukazwelonke. Ukucaciswa kwelungelo lobunikazi kukhombisa ukuthi i-10μM(micromol/L) ye-cepharanthine ivimbela ukuphindaphinda kwe-coronavirus ngesilinganiso esingu-15,393. .
Izinkambu zokufaka isicelo ze-cepharanthine
Isetshenziswa kwezokwelapha(COVID-19).
Amapharamitha womkhiqizo
IPHROFAYELA YENKAMPANI | |
Igama Lomkhiqizo | I-Cepharanthine |
CAS | 481-49-2 |
I-Chemical Formula | I-C37H38N2O6 |
Birandi | Hande |
Mumenzi | Inkampani Yunnan Hande Bio-Tech Co., Ltd. |
Cukuphuma | Kunming, China |
Imisiwe | 1993 |
BULWAZI LWE-ASIC | |
Omqondofana | 1H-4,6:16,19-Dietheno-21,25-metheno-12H-[1,3]dioxolo[4,5-g]pyrido[2',3':17,18][1,10] i-dioxacycloeicosino[2,3,4-ij]isoquinoline,2,3,13,14,14a,15,26,26a-octahydro-22,30-dimethoxy-1,14-dimethyl-,(14aS,26aR)-; I-Cepharanthine,>=98%;Cepharanthin,98%,fromStephaniajaponica(Thunb.)Miers;Cepharanthine|||CEPHARANTHINE;CEPHARANTHIN;CEPHARANTHIN;OXYACAANTHAN,6',12'-DIMETHOXY-2,2'-DIMETHYL-67, (METHYLLENEBIS(OXY))-;cepharantin |
Isakhiwo | |
Isisindo |
|
HIkhodi ye-S | N/A |
IkhwalithiSukucaciswa | Ukucaciswa Kwenkampani |
Cizitifiketi | N/A |
Isivivinyo | Kwenziwe ngokwezifiso ngokwezidingo zekhasimende |
Ukubukeka | Amakristalu amhlophe |
Indlela Yokukhipha | UStephania japonica (Thunb.) Miers |
Amandla Wonyaka | Kwenziwe ngokwezifiso ngokwezidingo zekhasimende |
Iphakheji | Kwenziwe ngokwezifiso ngokwezidingo zekhasimende |
Indlela Yokuhlola | I-HPLC |
Logistics | Izinto zokuthutha eziningi |
PaymentTerms | T/T, D/P, D/A |
Olapho | Yamukela ukuhlolwa kwamakhasimende ngaso sonke isikhathi;Siza amaklayenti ngokubhaliswa kokulawula. |
Isitatimende somkhiqizo we-Hande:
1. Yonke imikhiqizo ethengiswa yinkampani iyimpahla yokusetshenziswa engaqediwe.Imikhiqizo iqondiswe kakhulu kubakhiqizi abaneziqu zokukhiqiza, futhi izinto ezingavuthiwe aziyona imikhiqizo yokugcina.
2. Ukusebenza okungaba khona kanye nezicelo ezihilelekile esingenisweni konke kuvela ezincwadini ezishicilelwe.Abantu ngabanye abancomi ukusetshenziswa okuqondile, futhi ukuthenga ngakunye kwenqatshwa.
3. Izithombe nolwazi lomkhiqizo kule sizindalwazi kungokwereferensi kuphela, futhi umkhiqizo wangempela yiwo oyosebenza.
Imboni yezandla:
I-Yunnan hande Biotechnology Co., Ltd., eyasungulwa ngo-Agasti 1993, iyibhizinisi lobuchwepheshe obuphezulu eligxile ocwaningweni nasekuthuthukisweni kwe-biotechnology.Ngemva kweminyaka yokuthuthuka, i-hande isungule uhlelo oluphelele lwekhwalithi, ilawula ikhwalithi yemikhiqizo ngokuvumelana namazinga aphezulu, futhi yandisa inani lokukhipha amandla okukhiqiza.Imikhiqizo yayo isiphasise isitifiketi semithetho neziqondiso zamazwe ngamazwe, futhi ibe umkhiqizi wezitshalo ezingavuthiwe okwenza wonke umuntu azizwe ekhululekile.
Iba umphakeli ongcono kakhulu wezinto ezingavuthiwe namabhizinisi ngobuqotho!
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