Ulwazi Lomkhiqizo
Igama:Huperzine A
Inombolo ye-CAS:102518-79-6
Ifomula ye-molecular:I-C15H18N2O
Isakhiwo samangqamuzana:
Ukucaciswa:≥98%
Indlela yokuthola:I-HPLC
Umbala:i-crystalline powder ephuzi
Imiphumela ye-Pharmacological ye-huperzine A
I-Huperzine A iyi-inhibitor ye-cholinesterase eguqulekayo esebenza kahle kakhulu enomsebenzi oqinile we-cholinergic.Ekuqaleni yayisetshenziselwa ukwelapha i-myasthenia gravis.Ngemva kokubhekwa komtholampilo, inomphumela obalulekile wokuthuthukisa inkumbulo kubantu asebekhulile abanokukhubazeka kwenkumbulo okuhle futhi ingathuthukisa inkumbulo nemisebenzi yengqondo.I-Pharmacological ukuhlola kubonise ukuthi i-huperzine A inomsebenzi oqinile we-cholinergic kanye nokuvinjelwa okukhethiwe okuguquguqukayo ku-cholinesterase yangempela.Ingenza kube lula ukudluliswa kwama-neurotransmitters endaweni ye-neuromuscular junction.Ingakhuphula kakhulu izinga le-acetylcholine, ikhuthaze ukubuyiswa kwenkumbulo futhi ithuthukise inkumbulo.
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