I-Cabazitaxel Cas 183133-96-2 Umkhiqizi we-Cabazitaxil

Incazelo emfushane:

I-Carbataxel iyikhemikhali esetshenziselwa ukwenza izidakamizwa ezilwa nomdlavuza.I-Carbataxel iyimpushana emhlophe noma emhlophe ecishe ingancibiliki emanzini, kodwa inyibilika ku-ethanol.Indlela yayo yokulwa nomdlavuza nezici ziyafana ne-docetaxel, futhi ingeyesigaba semithi elwa ne-microtubule.Ngokusebenzisa hlanganisa ne tubulin, ukhuthaze ukuhlangana yayo zibe microtubules, ngasikhathi sinye kungavimbela lezi uye wabutha microtubule disassembly, ukuthi ukuzinza microtubules, ngaleyo ndlela inhibite cell mitosis, kanye interphase cell function (interphasecellularfunctions).


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Ulwazi Lomkhiqizo

Igama:I-Cabazitaxel

Inombolo ye-CAS:183133-96-2

Ifomula yekhemikhali:I-C45H57NO14

Imininingwane:99%

Umbala:impushana emhlophe noma emhlophe

Umthombo:Ihlanganiswe kancane ne-10-DAB

Uhlobo:Ama-API

Umphumela

I-Carbataxel iwukuphuma kwe-taxane esebenza njenge-microtubule inhibitor, ebophezela ku-tubulin futhi ithuthukise ukuhlangana kwayo kuma-microtubules, kuyilapho ivimbela ukuhlakazeka kwalawa ma-microtubules ahlanganisiwe futhi kusimamisa ama-microtubules.Lokhu kuvimbela kubangela ukuhlukaniswa kwama-microtubules kanye nokuyeka ukuhlukana kwamaseli, ngaleyo ndlela kumise umjikelezo wamangqamuzana futhi kuvimbele ukwanda kwesimila.Ngakho-ke, i-carbataxel isetshenziselwa ikakhulukazi ukulungiswa kwezidakamizwa ezilwa nomdlavuza, inomphumela omuhle wokulwa nomdlavuza, futhi ingasetshenziswa ukwelapha izifo ezihlukahlukene zamagciwane.Ngokucacile, i-carbataxel isetshenziswe kabanzi ukwelapha i-prostate, ibele, i-ovarian, i-lung, kanye nezinye izinhlobo eziningi zomdlavuza, kanye nokutheleleka kwamagciwane, okuhlanganisa i-sinusitis, i-bronchitis, i-pneumonia, izifo ze-urinary tract, izifo zamehlo, izifo zesikhumba, ne-otitis media.

Izinkonzo Zethu

1.Imikhiqizo:Nikeza ngezingcaphuno zezitshalo zekhwalithi ephezulu, ezihlanzeke kakhulu, izinto zokusetshenziswa zemithi, nezimaphakathi zemithi.

2.Izinsizakalo zobuchwepheshe:Izingcaphuno ezenziwe ngokwezifiso ezinemininingwane ekhethekile ngokuya ngezidingo zekhasimende.

Imboni yezandla

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