I-paclitaxel yemvelo ye-paclitaxel apis imithi ye-anticancer apis

Incazelo emfushane:

I-Natural paclitaxel iyinhlanganisela yemvelo ebalulekile ekhishwe egxolweni le- taxus chinensis.Kuyisidakamizwa semvelo esilwa nomdlavuza futhi sisetshenziswa kakhulu ekwelapheni izimila eziyingozi njengomdlavuza webele, umdlavuza wamaphaphu kanye nomdlavuza wesisu.Uma kuqhathaniswa nezinye izidakamizwa ezilwa nomdlavuza, i-paclitaxel yemvelo inephrofayili yokuphepha ephezulu kanye nemiphumela engemihle embalwa.


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Ulwazi Lomkhiqizo

Igama:I-Paclitaxel

Inombolo ye-CAS:33069-62-4

Ifomula yekhemikhali:I-C47H51NO14

Imininingwane:99%-102%

Umbala:impushana emhlophe noma ecishe ibe mhlophe

Umthombo:I-Taxus yunnanensis, i-Taxus chinensis

Uhlobo:Ama-API

Indima ye-paclitaxel yemvelo

I-1, ivimbela ukuhlukana kwe-tumor cell kanye nokusabalala: i-paclitaxel yemvelo ingaphazamisa inqubo yokuhlukaniswa kwamangqamuzana nokwanda, okuholela ekutheni amangqamuzana omdlavuza angakwazi ukukhula nokuzala ngokujwayelekile, ngaleyo ndlela avimbele ukuthuthukiswa nokusabalala kwamathumba.

2, bangela i-tumor cell apoptosis: I-paclitaxel yemvelo ingabangela inqubo yokuzilimaza ebangela ukuthi amangqamuzana omdlavuza azifele ngokwawo, eyaziwa ngokuthi i-apoptosis.Le ndlela ingabulala ngempumelelo amangqamuzana omdlavuza, inciphise umthamo wesimila, futhi ikhulule izimpawu zeziguli.

3. Vimbela i-angiogenesis yesimila: ukukhula nokusabalala kwamathumba kudinga imithambo yegazi emisha ukuze inikeze imisoco.I-paclitaxel yemvelo ingavimbela umsebenzi we-vascular endothelial growth factor, ngaleyo ndlela ivimbele ukwakheka kwemithambo yegazi yesimila, inqamule ukunikezwa kwezakhi zamathumba, futhi kuholele ekufeni kwamaseli wesimila.

Izinkonzo Zethu

1.Imikhiqizo:Nikeza ngezingcaphuno zezitshalo zekhwalithi ephezulu, ezihlanzeke kakhulu, izinto zokusetshenziswa zemithi, nezimaphakathi zemithi.

2.Izinsizakalo zobuchwepheshe:Izingcaphuno ezenziwe ngokwezifiso ezinemininingwane ekhethekile ngokuya ngezidingo zekhasimende.

Imboni yezandla

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